JPH0122264B2 - - Google Patents

Info

Publication number
JPH0122264B2
JPH0122264B2 JP55137512A JP13751280A JPH0122264B2 JP H0122264 B2 JPH0122264 B2 JP H0122264B2 JP 55137512 A JP55137512 A JP 55137512A JP 13751280 A JP13751280 A JP 13751280A JP H0122264 B2 JPH0122264 B2 JP H0122264B2
Authority
JP
Japan
Prior art keywords
formula
general formula
heterocyclic amine
pyrrolidinyl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP55137512A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5649351A (en
Inventor
Tomine Misheru
Furanseshiinu Jakuriinu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ECHUUDO SHIANTEIFUIKU E IND DO RIRU DO FURANSU SOC
Original Assignee
ECHUUDO SHIANTEIFUIKU E IND DO RIRU DO FURANSU SOC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7917610A external-priority patent/FR2460935A1/fr
Priority claimed from FR8007352A external-priority patent/FR2479218A2/fr
Application filed by ECHUUDO SHIANTEIFUIKU E IND DO RIRU DO FURANSU SOC filed Critical ECHUUDO SHIANTEIFUIKU E IND DO RIRU DO FURANSU SOC
Publication of JPS5649351A publication Critical patent/JPS5649351A/ja
Publication of JPH0122264B2 publication Critical patent/JPH0122264B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/08—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP13751280A 1979-07-06 1980-09-30 Heterocyclic amine and its manufacture Granted JPS5649351A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7917610A FR2460935A1 (fr) 1979-07-06 1979-07-06 Nouvelles phenoxyamines heterocycliques substituees, leur methode de preparation et leur application comme anesthetiques locaux
FR8007352A FR2479218A2 (fr) 1980-04-01 1980-04-01 Nouvelles phenoxyamines heterocycliques substituees, leur methode de preparation et leur application comme anesthesiques locaux

Publications (2)

Publication Number Publication Date
JPS5649351A JPS5649351A (en) 1981-05-02
JPH0122264B2 true JPH0122264B2 (en]) 1989-04-25

Family

ID=26221244

Family Applications (2)

Application Number Title Priority Date Filing Date
JP9321680A Granted JPS5639065A (en) 1979-07-06 1980-07-07 Novel phenoxy heterocyclic amine* its manufacture and local narcotic as active component thereof
JP13751280A Granted JPS5649351A (en) 1979-07-06 1980-09-30 Heterocyclic amine and its manufacture

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP9321680A Granted JPS5639065A (en) 1979-07-06 1980-07-07 Novel phenoxy heterocyclic amine* its manufacture and local narcotic as active component thereof

Country Status (37)

Country Link
US (1) US4379161A (en])
EP (2) EP0024960B1 (en])
JP (2) JPS5639065A (en])
AR (1) AR224012A1 (en])
AT (2) ATE10739T1 (en])
AU (2) AU536482B2 (en])
BE (1) BE884124A (en])
BG (2) BG35039A3 (en])
CA (1) CA1163273A (en])
CH (2) CH648827A5 (en])
CS (1) CS216933B2 (en])
DD (2) DD201141A5 (en])
DE (2) DE3069789D1 (en])
DK (1) DK157538C (en])
ES (1) ES493111A0 (en])
FI (2) FI872955A7 (en])
GR (1) GR69638B (en])
HK (2) HK55889A (en])
HU (2) HU181147B (en])
IE (2) IE50061B1 (en])
IL (2) IL60472A (en])
IN (2) IN153037B (en])
IT (1) IT1188985B (en])
JO (1) JO1077B1 (en])
LU (1) LU82584A1 (en])
MA (1) MA18893A1 (en])
MX (2) MX7642E (en])
NO (2) NO156086C (en])
NZ (1) NZ194230A (en])
OA (1) OA06561A (en])
PH (1) PH16449A (en])
PL (1) PL127393B1 (en])
PT (1) PT71482A (en])
RO (2) RO85323B (en])
SU (1) SU1085507A3 (en])
YU (2) YU42344B (en])
ZW (1) ZW15280A1 (en])

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2586018B1 (fr) * 1985-08-12 1988-03-25 Ile De France Nouveau benzodioxepanne, son procede de synthese et ses applications en therapeutique
WO1990012004A1 (en) * 1989-04-07 1990-10-18 Fujisawa Pharmaceutical Co., Ltd. New naphthalene compounds and method of producing the same
EP0471941A3 (en) * 1990-08-16 1992-10-14 American Cyanamid Company An improved process for the preparation of 5-bromo-2-methoxyresorcinol
US5472958A (en) * 1994-08-29 1995-12-05 Abbott Laboratories 2-((nitro)phenoxymethyl) heterocyclic compounds that enhance cognitive function
US7799337B2 (en) * 1997-07-21 2010-09-21 Levin Bruce H Method for directed intranasal administration of a composition
ATE247104T1 (de) * 1997-11-05 2003-08-15 Neurosearch As Azaring-ether-derivate und ihre verwendung als nicotinic-ach-rezeptormodulatoren
US8473062B2 (en) * 2008-05-01 2013-06-25 Autonomic Technologies, Inc. Method and device for the treatment of headache
US8412336B2 (en) 2008-12-29 2013-04-02 Autonomic Technologies, Inc. Integrated delivery and visualization tool for a neuromodulation system
US8494641B2 (en) 2009-04-22 2013-07-23 Autonomic Technologies, Inc. Implantable neurostimulator with integral hermetic electronic enclosure, circuit substrate, monolithic feed-through, lead assembly and anchoring mechanism
US9320908B2 (en) * 2009-01-15 2016-04-26 Autonomic Technologies, Inc. Approval per use implanted neurostimulator
US20100185249A1 (en) * 2009-01-22 2010-07-22 Wingeier Brett M Method and Devices for Adrenal Stimulation
CN111205015B (zh) * 2020-01-20 2021-11-26 东南大学 一种高稳定泡沫混凝土发泡剂的制备方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE543876C (de) * 1928-04-25 1932-02-11 C H Boehringer Sohn Akt Ges Verfahren zur Darstellung von Piperidinalkinen
US3117976A (en) * 1958-11-12 1964-01-14 Beecham Res Lab Nu-alkyl-pyrrolidine-2-methanol, alpha cyclohexyl mandelates
FR1342756A (fr) * 1958-11-21 1963-11-15 Beecham Res Lab Esters basiques et leur procédé de préparation, notamment le phényl-cyclohexyl-glycolate de (1-méthyl-2-pyrrolidyl) méthyle et ses sels d'addition
GB1096441A (en) * 1964-01-15 1967-12-29 Bristol Myers Co Ethers of benzyl phenols and a process for the preparation thereof
US3904622A (en) * 1968-02-16 1975-09-09 Ile De France Dialkylaminoalkyl ethers of 2-alkoxy-3,5-dihalobenzene
GB1268951A (en) * 1969-06-12 1972-03-29 Pfizer Ltd Phenoxy-amines
FR2155927A1 (en) * 1971-10-15 1973-05-25 Synthelabo 1-phenylcyclo hexane carboxylic acid esters - with antispasmodic and anticholinergic activity
JPS5139661A (en) * 1974-09-27 1976-04-02 Nippon Kayaku Kk Kogakukatsusei 11 mechiru 22 * beetaaa hidorokishechiru * pirorijin oyobisono chukantaino seizoho
JPS5251362A (en) * 1975-10-20 1977-04-25 Teijin Ltd Preparation of optically active pyrrolidine derivatives
LU78625A1 (de) * 1977-12-02 1979-06-13 Byk Gulden Lomberg Chem Fab Substituierte 1-phenyl-2-pyrrolidin-2-yl-ethanole,verfahren zu ihrer herstellung,ihre verwendung und sie enthaltende arzneimittel
DE2811952A1 (de) * 1978-03-18 1979-10-31 Merck Patent Gmbh Phenoxyalkylamine und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
PL225473A1 (en]) 1981-10-16
DD153206A5 (de) 1981-12-30
NO802027L (no) 1981-01-07
IN158706B (en]) 1987-01-10
HK55689A (en) 1989-07-21
YU42824B (en) 1988-12-31
DK289580A (da) 1981-01-07
BE884124A (fr) 1981-01-05
IT8049163A0 (it) 1980-07-04
MX7642E (es) 1990-05-16
BG35039A3 (bg) 1984-01-16
GR69638B (en]) 1982-07-06
IE801392L (en) 1981-01-06
SU1085507A3 (ru) 1984-04-07
IN153037B (en]) 1984-05-26
PT71482A (fr) 1980-08-01
YU171080A (en) 1983-06-30
AU536482B2 (en) 1984-05-10
FI74274B (fi) 1987-09-30
JO1077B1 (en) 1982-07-10
IL60472A0 (en) 1980-09-16
FI872955A0 (fi) 1987-07-03
ATE17119T1 (de) 1986-01-15
ES8103049A1 (es) 1981-02-16
RO85323A (ro) 1984-09-29
DE3071314D1 (en) 1986-02-06
CH655100A5 (fr) 1986-03-27
MA18893A1 (fr) 1981-04-01
NO156086C (no) 1987-07-22
EP0094102A2 (fr) 1983-11-16
FI74274C (fi) 1988-01-11
EP0094102B1 (fr) 1985-12-27
US4379161A (en) 1983-04-05
RO81532B (ro) 1983-04-30
FI872955L (fi) 1987-07-03
IT1188985B (it) 1988-01-28
IE801390L (en) 1981-01-04
AR224012A1 (es) 1981-10-15
IT8049163A1 (it) 1982-01-04
NZ194230A (en) 1983-02-15
NO156086B (no) 1987-04-13
AU6002880A (en) 1981-01-15
OA06561A (fr) 1981-07-31
CH648827A5 (fr) 1985-04-15
AU563009B2 (en) 1987-06-25
PL127393B1 (en) 1983-10-31
ES493111A0 (es) 1981-02-16
AU2526084A (en) 1984-07-26
LU82584A1 (fr) 1981-02-02
RO85323B (ro) 1984-10-30
BG35746A3 (bg) 1984-06-15
EP0024960A3 (en) 1981-06-17
YU280182A (en) 1983-06-30
JPS5639065A (en) 1981-04-14
EP0024960B1 (fr) 1984-12-12
IL68854A0 (en) 1983-10-31
ZW15280A1 (en) 1980-10-01
HU186539B (en) 1985-08-28
CA1163273A (fr) 1984-03-06
HK55889A (en) 1989-07-21
JPS5649351A (en) 1981-05-02
DK157538C (da) 1990-06-11
DD201141A5 (de) 1983-07-06
DE3069789D1 (en) 1985-01-24
CS216933B2 (en) 1982-12-31
ATE10739T1 (de) 1984-12-15
PH16449A (en) 1983-10-12
YU42344B (en) 1988-08-31
EP0024960A2 (fr) 1981-03-11
DK157538B (da) 1990-01-22
NO861988L (no) 1981-01-07
IE50060B1 (en) 1986-02-05
IE50061B1 (en) 1986-02-05
EP0094102A3 (en) 1984-04-11
JPH0149704B2 (en]) 1989-10-25
HU181147B (en) 1983-06-28
MX6366E (es) 1985-05-21
IL60472A (en) 1983-09-30
FI802156A7 (fi) 1981-01-07
RO81532A (ro) 1983-04-29
FI872955A7 (fi) 1987-07-03

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